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Search Results for " cdk4/6 inhibitor iv "

2

Compounds

Cat No. Product Name Synonyms Targets
T21720 GP-82996 Cdk4/6 Inhibitor IV,CINK4 CDK
GP-82996 (CINK4) is a pharmacological inhibitor specifically targeting CDK4/6, exhibiting IC50 values of 1.5 μM for CDK4/cyclin D1, 5.6 μM for CDK6/cyclin D1, and 25 μM for Cdk5/p35. It effectively induces apoptosis in U...
T36967 LSN3106729 hydrochloride
LSN3106729 hydrochloride, the metabolite of Abemaciclib , is a CDK inhibitor with antitumor activity. LSN3106729 hydrochloride and a CRBN ligand have been used to design PROTAC CDK4/6 degrader[1]. [1]. Edward S. Kim, et ...
TargetMol